Proviron is the Schering brand name for the oral androgen mesterolone. It is a strong androgen, which is not capable of aromatizing into estrogen. It is also not progestenic.
In fact, Proviron is the closest thing we have to orally active Dihydrotestosterone (DHT).
Physicians normally prescribe this compound to treat various types of sexual dysfunction since it can usually reverse impotency and sexual disinterest. It can also increase sperm count although it does not actually stimulate testosterone production.

In bodybuilding circles, Proviron is used primarily as an anti-estrogen since it is believed to block the action of the aromatase enzyme (which is responsible for converting testosterone to estrogen). For this reason it is a popular pre-contest drug since it assists in hardening up the physique.

Whilst Proviron is considered too weak for muscle building purposes it may actually boost the anabolic effect of other substances when it is added to a standard cycle. This is due to the fact that it binds to Sex Hormone Binding Globulin (SHBG), which is the transport hormone responsible for reducing the amount of free testosterone in your body. In addition to this, Proviron also binds to the Anabolic Receptor more effectively than any other oral steroid. So, not only does Proviron reduce levels of circulating estrogen, it can possibly make other steroids more effective through its ability to inhibit the actions of SHBG. It is also worth pointing out that even at levels of 100-150mg/day it has no depressing effect on low to normal FSH (Follicle Stimulating Hormone) and LH (Luteinizing Hormone) levels. In fact it has been suggested that it may even raise LH, which can in turn lead to a rise in testosterone levels.

DOSAGE

The typical dosage for men is one to four 25mg tablets per day. This is considered to be a sufficient amount to avoid the occurrence of gynecomastia. It may also be combined with Nolvadex (tamoxifen citrate) or Clomid (clomiphene citrate) when substances with high estrogenic conversion rates are being taken (e.g. Dianabol, Testosterone). In this instance, taking 50mg of Proviron along with 20mg Nolvadex per day has been proven effective.

In the case of women considering using Proviron it has to be noted that it does have an extremely high androgen content. With this in mind care should be taken when it comes to assessing dosages. Women usually find 25mg per day is enough to effectively shift the androgen/estrogen level, which can have a significant impact on the physique. Also, in order to avoid virilization symptoms (e.g. voice deepening, menstrual irregularities, skin texture changes, clitoral enlargement) use should be limited to a period of four or five weeks.

Once again, a combination of 25mg Proviron and 10-20mg Nolvadex can be very efficient when it comes to muscle hardening and ridding the body of extra body fat on hips and thighs.

SAFETY ISSUES

The risk of liver toxicity with this compound is generally not an issue since Proviron is not a c17 alpha alkylated compound (the alteration responsible for liver toxicity in commonly used anabolics). It is therefore considered to be a ‘safe’ oral.

However, that does not mean that is comes without side effects. In the case of male athletes using this drug in amounts above 100mg a day side effects connected with an excessively high androgen level can present themselves. These include oily skin, acne, body/facial hair growth, and male pattern baldness. Extreme heightening of the male libido is also likely.

As previously mentioned, women should be careful when using this substance and stick to 25mg a day for short periods of time to avoid virilization symptoms.

In addition, since Proviron is a very effective ‘drying agent’ it can also have a significant impact on the condition of your hair and skin. It is therefore recommended that an essential fatty acid supplement be used with this product, which supplies the omega 3 fats necessary to maintain healthy skin and hair. Also, as a DHT derivative thinning hair may be a problem in susceptible individuals. In this instance some have found the use of Nizoral shampoo to be of assistance.

Leigh Penman, in addition to be a staff writer at MuscleSport Mag, has been writing for bodybuilding magazines, websites and nutritional supplement companies since 1985. Whilst residing in the UK, she earned the reputation of being one of the top female writers in bodybuilding-related media. Her credits included being a contributing editor on all the magazines in production as well as filling the shoes of Ladies Editor and Showbiz Editor on two publications (the later being on Arnold’s sanctioned magazine, ‘Bodypower’). During this time she also competed successfully on four occasions (placing in the top four in all contests).

Leigh has been working out for close to thirty years so she is clearly a writer who ‘walks her talk.’
She can be contacted personally at zeal2heal@yahoo.com or you can also check her out at New York’s favorite metaphysical store www.stickstoneandbone.com.

This is part of a continuing series provided exclusively by MuscleSport Mag giving information on a variety of performance-enhancing drugs for educational purposes. While it is apparent that people are going to use these substances regardless of the health and legal risks involved, quality information is necessary and learning as much about them as possible can only assist an adult making a decision either way.

Until fairly recently the mere suggestion of using the essentially male hormone testosterone to treat female patients would have been considered out of the question by the majority of the medical profession. However, with leading pharmaceutical company Procter & Gamble announcing the development of Intrinsa ( a testosterone patch for women who have gone through menopause after surgical removal of their ovaries and uterus) it seems that the times they are a changing!

The patch – which produces a 50 to 70 percent increase in sexual desire according to studies – is already available on prescription in the UK and, although it is only given to women who have had hysterectomies, it does mark an important change in the way we approach hormone therapy. In fact there are probably a large amount of women who would benefit greatly from treatment with therapeutic doses of testosterone since,even before menopause occurs, many women have significantly lower levels of free testosterone (or any of its precursors such as DHEA). Additionally, in the years following menopause the levels are further reduced, leading to symptoms such as lack of libido, depression, fatigue and difficulty losing weight. When testosterone is administered the results can be quite dramatic with renewed outlook and enthusiasm for life, increased energy levels, reduction in fatigue, restoration of sex drive and greater ability to lose weight when following exercise and diet programs.

TESTOSTERONE AND WEIGHT LOSS

It is a simple fact of life that during the years preceding menopause and the years that follow, women experience changes in body composition – with noticeable increases in fat storage. This change in body composition can begin up to fifteen years before true menopause actually occurs. The hormone connection with this body composition alteration is rarely explored and, to make matters even worse, this is also the time when most doctors willingly distribute estrogens and progestins in the name of Hormone Replacement Therapy. This practice only serves to make matters worse since administering estrogen and progesterone makes it almost impossible for a woman to lose weight. After all, isn’t estrogen used by farmers to fatten up livestock swiftly and increase their turnover/profit margins? Any woman who has used birth control pills during her lifetime will attest to the fact that weight gain is usually a side effect of their use – from as little as 3 pounds to as much as 8-10 pounds being
experienced.

So where does testosterone come into the equation?
Well, it is a widely held belief that testosterone causes weight gain, since studies have been published linking abdominal obesity with elevated testosterone levels in women. The flaw in this conclusion is the ‘conveniently omitted’ discovery that these women not only have elevated testosterone levels but their whole hormone profile is out of balance and, in addition, their insulin levels are high with poor insulin sensitivity – a well reported culprit in the cause of obesity. However, even the mere suggestion that testosterone administration may be beneficial for some women is taboo and the facilitation of studies to explore this rubs shoulders with the concept of studying the possibilities of male childbirth (although recent news reports point to even this possibility being currently explored – albeit in a transgender individual).

There have been trials conducted on a transdermal testosterone gel for women which would allow for a slow release of testosterone into the bloodstream, keeping levels elevated for about six hours and bypassing the liver. This substance has received little media attention though and has, for the best part, taken up residence on the shelf occupied by other drugs, which are either considered inappropriate or unsafe for use.

TESTOSTERONE AND SEXUAL DYSFUNCTION

Libido is another area where testosterone plays a major role in women where sexual dysfunction is often caused by a low interest in sex. Administering testosterone in such cases has often restored women’s sex drives to youthful levels with increases in the ability to achieve orgasm as well as length of orgasm experienced. Needless to say, the increased interest and participation in sexual activity significantly relieves stress and depression as well as improving the quality of relationships and favorably influencing body composition via the increased energy expenditure involved.

THE SIDE EFFECTS

Of course it would be totally irresponsible to neglect to mention the side effects which may be experienced by women introducing testosterone to their system. After all, you are introducing an essentially male hormone into a female body. Of course, side effects are also substance (which form of testosterone used) and dose related but they do include such things as:

* Hirsutism (increased hair growth on face, chest, around nipples and buttocks.)

* Deepening of the voice – beginning with hoarseness before the voice actually ‘breaks’ like that of a pubescent male.

* Vaginal Discharge can sometimes present itself. This is not a sign of infection but if it occurs -which is not always the case – can be troublesome.

* Clitoral Enlargement – which may or may not be considered a negative effect (depending on the amount of ‘growth’ involved). It does however usually lead to a greater frequency and intensity of orgasms.

* Menstrual Irregularities or amenorrhea (absence of menstrual cycle for six months or more). Of course this is not of concern to postmenopausal women and may even be considered an asset by pre-menopausal women.

Wrapping up the side effects issue, it has to be said that the onset of virilization symptoms (deepening of the voice, increased body and facial hair growth, acne etc) can differ greatly between women depending on individual sensitivities and genetics. It is therefore advised that a female considering testosterone use should start by using low dosages (even a testosterone pro-hormone) and carefully monitoring effects. Also keeping cycles short allowing for sufficient breaks in administration.

TESTOSTERONE THERAPY

In conclusion, perhaps the time is coming where testosterone will actually be considered as a therapeutic agent when it comes to treating both pre and post menopausal women. It certainly beats the current standard of loading them up with estrogen (which often leads to increased fat mass and loss of muscle).
If you are suffering from any of the previously mentioned symptoms of low testosterone you are advised to consult a physician in order to obtain a complete hormone profile. From there you can decide whether hormone therapy is for you or if the addition of some of the over the counter food supplements would be of value.
Testosterone and progesterone levels can often be restored by natural means and once this natural balance is restored women often find it easier to reach their weight loss goals and can reverse the loss of muscle and bone mass that occurs with age.

NATURAL STEPS TO TESTOSTERONE BOOSTING

There are many steps that can be taken to naturally enhance the production of testosterone and these include:

* Increasing your intake of testosterone-boosting protein foods. These foods include lean cuts of beef, eggs, chicken and turkey breasts, cottage cheese and oysters. You should consume at least 1 gram of protein per pound of bodyweight each day.

* Eat testosterone-boosting vegetables such as broccoli, cabbage and Brussels sprouts. These vegetables are high in indoles, which increase testosterone by reducing the estrogenic effects of estradiol (a form of estrogen known to inhibit testosterone).

* Add saturated fats to your diet. This is not an invitation to pig out at MacDonald’s but it is important to have a sufficient amount of dietary fat in your diet to facilitate testosterone production. Aim for a healthy mix of saturated and unsaturated fats (about 50/50) and try to get about 4 calories per pound of bodyweight from dietary fat. For a 150lb athlete this would amount to 600 calories from fat – about 66 grams a day.

* Do not restrict calories too drastically. Low calorie intakes are notorious for killing testosterone. Unless you are on a pre contest regime, try to get at least 16-18 calories for each pound of bodyweight.

WOMEN AND TESTOSTERONE…THE FUTURE

The whole purpose of this article is to throw a new perspective on hormone therapy under the spotlight. Perhaps the time has come to bury the old ‘pink for girls, blue for boys’ theory of hormone replacement and put some research into testosterone therapy when it comes to helping women lead fuller lives.

It is certainly a controversial subject, but it is also thought provoking and definitely worthy of further investigation. What’s more, I am sure we will hear much more about this form of hormone therapy in the future as the results of existing studies begin to filter their way into the mainstream media.

Leigh Penman, in addition to be a staff writer at MuscleSport Mag, has been writing for bodybuilding magazines, websites and nutritional supplement companies since 1985. Whilst residing in the UK, she earned the reputation of being one of the top female writers in bodybuilding-related media. Her credits included being a contributing editor on all the magazines in production as well as filling the shoes of Ladies Editor and Showbiz Editor on two publications (the later being on Arnold’s sanctioned magazine, ‘Bodypower’). During this time she also competed successfully on four occasions (placing in the top four in all contests).

Relocating to New York in the late 1990s she focused her writing attention to crystal healing techniques and metaphysics – however, she still maintained a five day workout schedule during this time and gained her personal training certificate.

Leigh has been working out for close to thirty years so she is clearly a writer who ‘walks her talk.’
She can be contacted personally at zeal2heal@yahoo.com or you can also check her out at New York’s favorite metaphysical store www.stickstoneandbone.com.